SCHEMBL2904593

SCHEMBL2904593

CCOC(=O)c1cnc2cc(OC)c(Br)cc2c1Nc1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.64
CSF1R P07333 3/20 0.63
GAA P10253 4/20 0.60
THRB P10828 2/20 0.60
TP53 P04637 3/20 0.57
SMN1; SMN2 Q16637 4/20 0.56
ALDH1A1 P00352 1/20 0.56
HTT P42858 1/20 0.56
PAX8 Q06710 1/20 0.55
EGFR P00533 1/20 0.52
MEN1 O00255 1/20 0.51
SLC2A1 P11166 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4081004 0.91 MAPT (0.58) MAPTCSF1RGAATHRBTP53
SCHEMBL2913279 0.91 CSF1R (0.64) MAPTCSF1RGAATHRBTP53
SCHEMBL23575246 0.90 MAPT (0.61) MAPTGAATHRBTP53SMN1; SMN2
SCHEMBL2912196 0.89 CSF1R (0.64) MAPTCSF1RGAATHRBTP53
SCHEMBL2909819 0.88 MAPT (0.72) MAPTCSF1RGAATHRBTP53
SCHEMBL2905486 0.88 MAPT (0.67) MAPTCSF1RGAATHRBMEN1
SCHEMBL2908163 0.87 CSF1R (0.64) MAPTCSF1RGAATHRBTP53
SCHEMBL2913350 0.84 MAPT (0.59) MAPTGAATHRBTP53SMN1; SMN2
SCHEMBL2910297 0.84 MAPT (0.59) MAPTCSF1RGAATHRBTP53
SCHEMBL2913881 0.84 CSF1R (0.65) MAPTCSF1RGAATHRBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed