SCHEMBL2912196

SCHEMBL2912196

CCOC(=O)c1cnc2cc(OC)c(Br)cc2c1Nc1ccc(F)c(F)c1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 3/20 0.64
MAPT P10636 8/20 0.58
TP53 P04637 3/20 0.58
EGFR P00533 1/20 0.55
GAA P10253 1/20 0.54
THRB P10828 1/20 0.54
CA2 P00918 1/20 0.53
NPSR1 Q6W5P4 2/20 0.52
LMNA P02545 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
PAX8 Q06710 1/20 0.52
AURKB Q96GD4 2/20 0.51
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
CLK1 P49759 1/20 0.51
AURKA O14965 1/20 0.50
POLB P06746 1/20 0.49
CREBBP Q92793 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2904593 0.89 MAPT (0.64) CSF1RMAPTTP53EGFRGAA
SCHEMBL4081004 0.88 MAPT (0.58) CSF1RMAPTTP53GAATHRB
SCHEMBL2913279 0.87 CSF1R (0.64) CSF1RMAPTTP53EGFRGAA
SCHEMBL23575246 0.87 MAPT (0.61) MAPTTP53EGFRGAATHRB
SCHEMBL2906337 0.86 CSF1R (0.66) CSF1RMAPTTP53GAATHRB
SCHEMBL2911260 0.86 CSF1R (0.65) CSF1RMAPTTP53GAATHRB
SCHEMBL2912397 0.85 CA2 (0.61) CSF1RMAPTTP53EGFRGAA
SCHEMBL2908274 0.85 CA2 (0.61) CSF1RMAPTTP53EGFRGAA
SCHEMBL2912047 0.85 CSF1R (0.64) CSF1RMAPTTP53GAATHRB
SCHEMBL2911907 0.84 CSF1R (0.66) CSF1RMAPTTP53GAATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed