SCHEMBL2904900

SCHEMBL2904900

CCOC(=O)c1ccc(N)c(S(C)(=O)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
MAOA P21397 1/20 0.54
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
CA12 O43570 2/20 0.51
CA7 P43166 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51
HPGD P15428 2/20 0.50
RECQL P46063 1/20 0.50
ALDH1A1 P00352 1/20 0.50
STS P08842 1/20 0.50
PTGER4 P35408 3/20 0.48
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
HCRTR1 O43613 1/20 0.47
HSD17B2 P37059 1/20 0.47
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911278 0.83 VCAM1 (0.56) LMNACYP1A2CA1CA2CA12
SCHEMBL14593012 0.82 ALDH1A1 (0.67) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL6471721 0.81 CA1 (0.72) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL30582428 0.80 LMNA (0.65) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL940578 0.80 LMNA (0.65) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL2913651 0.80 CA12 (0.50) CA1CA2CA12CA9CA14
SCHEMBL868290 0.79 LMNA (0.62) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL28740731 0.78 ALDH1A1 (0.49) CA1CA2CA12CA9CA14
SCHEMBL9879781 0.78 LMNA (0.53) LMNACYP1A2CYP3A4MAOACA1
SCHEMBL2896481 0.78 ALDH1A1 (0.62) LMNACYP1A2CYP3A4MAOACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4739682-A1 1,6-NAPHTHRIDINE COMPOUNDS AS SMARCA2 INHIBITORS USEFUL FOR THE TREATMENT OF SMARCA4 DEFICIENT CANCERS Janssen Pharmaceutica NV (BE) 2026-05-13 EP disclosed
WO-2025008058-A1 1,6-NAPHTHRIDINE COMPOUNDS AS SMARCA2 INHIBITORS USEFUL FOR THE TREATMENT OF SMARCA4 DEFICIENT CANCERS JANSSEN PHARMACEUTICA NV (BE) 2025-01-09 WO disclosed
EP-1325920-B1 N-SUBSTITUTED BENZOTHIOPHENESULFONAMIDE DERIVATIVES TOA EIYO LTD (JP) 2010-08-25 EP disclosed
US-7399781-B2 N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD. (JP) 2008-07-15 US disclosed
US-7071220-B2 N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD. (JP) 2006-07-04 US disclosed
US-20060116408-A1 N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD. (JP) 2006-06-01 US disclosed
CN-1245400-C N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD (JP) 2006-03-15 CN disclosed
US-20030229126-A1 N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD. 2003-12-11 US disclosed
CN-1458928-A N-substituted benzothiophenesulfonamide derivatives TOA EIYO LTD (JP) 2003-11-26 CN disclosed
EP-1325920-A1 N-SUBSTITUTED BENZOTHIOPHENESULFONAMIDE DERIVATIVES TOA EIYO LTD. (JP) 2003-07-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060116408-A1 N-substituted benzothiophenesulfonamide derivatives ECE1, ECE2, CMA1 LMNA 2757/4885CYP1A2 3621/4885CYP3A4 3905/4885
US-20030229126-A1 N-substituted benzothiophenesulfonamide derivatives ECE1, ECE2, CMA1 LMNA 2757/4885CYP1A2 3621/4885CYP3A4 3905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.