SCHEMBL290496

SCHEMBL290496

CC[n+]1ccccc1C(C)=O.O=S(=O)([O-])c1ccccc1

nearest known ligand 0.37

Known targets — ChEMBL curated mechanism

CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.37
PSIP1 O75475 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
BCAT1 P54687 1/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1712432 0.93 KDM4E (0.40) HSD11B1CYP2D6ALDH1A1KMT2AKDM4E
Sulfuric Acid SCHEMBL2183752 0.89 CYP2D6 (0.36) HSD11B1PSIP1L3MBTL1CYP2D6CYP2C19
Sulfuric Acid SCHEMBL1716752 0.89 CYP2D6 (0.36) HSD11B1PSIP1L3MBTL1CYP2D6CYP2C19
SCHEMBL290641 0.87 CYP2D6 (0.35) HSD11B1PSIP1L3MBTL1CYP2D6CYP2C19
SCHEMBL1650870 0.86 CYP2D6 (0.35) HSD11B1PSIP1L3MBTL1CYP2D6CYP2C19
SCHEMBL1716087 0.86 CYP2D6 (0.54) L3MBTL1CYP2D6CYP2C19ALDH1A1KMT2A
SCHEMBL1724143 0.86 CYP2D6 (0.41) HSD11B1CYP2D6CYP2C19ALDH1A1KMT2A
SCHEMBL1712336 0.85 L3MBTL1 (0.34) HSD11B1PSIP1L3MBTL1CYP2D6CYP2C19
Acetic Acid SCHEMBL1712859 0.84 CYP2D6 (0.38) CYP2D6CYP2C19ALDH1A1GAAKMT2A
Bromide SCHEMBL1712146 0.84 CYP2D6 (0.40) CYP2D6CYP2C19ALDH1A1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2263642-B1 Colouring bleaches HENKEL AG & CO KGAA (DE) 2020-04-15 EP disclosed
EP-2427247-A2 FOIL APPLICATOR Henkel AG & Co. KGaA (DE) 2012-03-14 EP disclosed
EP-2320854-B1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES HENKEL AG & CO KGAA (DE) 2012-01-18 EP disclosed
US-8034122-B2 Bleaching agent comprising 2-acylpyridinium derivatives HENKEL AG & CO. KGAA (DE) 2011-10-11 US disclosed
EP-2344113-A2 MEANS FOR TREATING KERATIN FIBRES CONTAINING CATIONIC PYRIDINIUM DERIVATIVES Henkel AG & Co. KGaA (DE) 2011-07-20 EP disclosed
US-20110162671-A1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES HENKEL AG & CO. KGAA (DE) 2011-07-07 US disclosed
EP-2320854-A2 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES Henkel AG & Co. KGaA (DE) 2011-05-18 EP disclosed
EP-2306963-A1 MATTING ADDITIVE FOR BLOND HAIR DYING Henkel AG & Co. KGaA (DE) 2011-04-13 EP disclosed
EP-2263642-A2 Colouring bleaches Henkel AG & Co. KGaA (DE) 2010-12-22 EP disclosed
WO-2010127902-A2 FOIL APPLICATOR HENKEL AG & CO. KGAA (DE) 2010-11-11 WO disclosed
WO-2010054981-A2 COMBINATION OF CATIONIC BLEACH ACTIVATORS AND DYES HENKEL AG & CO. KGAA (DE) 2010-05-20 WO disclosed
WO-2010029006-A2 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES HENKEL AG & CO. KGAA (DE) 2010-03-18 WO disclosed
WO-2010015441-A1 MATTING ADDITIVE FOR BLOND HAIR DYING HENKEL AG & CO. KGAA (DE) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110162671-A1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES KRT18, CBR3, ACOX3 HSD11B1 2678/4885PSIP1 4615/4885L3MBTL1 3565/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.