SCHEMBL290641

SCHEMBL290641

CC(=O)C[n+]1ccccc1C(C)=O.O=S(=O)([O-])c1ccccc1

nearest known ligand 0.35

Known targets — ChEMBL curated mechanism

CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HSD11B1 P28845 2/20 0.33
KMT2A Q03164 2/20 0.33
LMNA P02545 2/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
BCAT1 P54687 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
PSIP1 O75475 1/20 0.33
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
ACHE P22303 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL143689 0.93 LMNA (0.38) CYP2D6HSD11B1KMT2ALMNAKDM4E
Sulfuric Acid SCHEMBL2182781 0.90 CYP2C19 (0.35) CYP2D6CYP2C19HSP90AA1KMT2ALMNA
Sulfuric Acid SCHEMBL291858 0.90 CYP2D6 (0.35) CYP2D6CYP2C19HSP90AA1KMT2ALMNA
SCHEMBL1712336 0.89 L3MBTL1 (0.34) CYP2D6CYP2C19HSP90AA1HSD11B1KMT2A
SCHEMBL290496 0.87 HSD11B1 (0.37) CYP2D6CYP2C19HSP90AA1HSD11B1KMT2A
SCHEMBL1723901 0.86 CYP2D6 (0.40) CYP2D6CYP2C19HSP90AA1KMT2ALMNA
Acetic Acid SCHEMBL1716728 0.85 CYP2C19 (0.37) CYP2D6CYP2C19KMT2ALMNAKDM4E
Bromide SCHEMBL1712392 0.85 CYP2D6 (0.39) CYP2D6CYP2C19KMT2ALMNAKDM4E
Hydrochloric Acid SCHEMBL1716730 0.85 CYP2D6 (0.39) CYP2D6CYP2C19HSP90AA1KMT2ALMNA
SCHEMBL1650870 0.84 CYP2D6 (0.35) CYP2D6CYP2C19HSP90AA1HSD11B1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427247-A2 FOIL APPLICATOR Henkel AG & Co. KGaA (DE) 2012-03-14 EP disclosed
EP-2320854-B1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES HENKEL AG & CO KGAA (DE) 2012-01-18 EP disclosed
US-8034122-B2 Bleaching agent comprising 2-acylpyridinium derivatives HENKEL AG & CO. KGAA (DE) 2011-10-11 US disclosed
EP-2344113-A2 MEANS FOR TREATING KERATIN FIBRES CONTAINING CATIONIC PYRIDINIUM DERIVATIVES Henkel AG & Co. KGaA (DE) 2011-07-20 EP disclosed
US-20110162671-A1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES HENKEL AG & CO. KGAA (DE) 2011-07-07 US disclosed
EP-2306963-A1 MATTING ADDITIVE FOR BLOND HAIR DYING Henkel AG & Co. KGaA (DE) 2011-04-13 EP disclosed
EP-2263642-A2 Colouring bleaches Henkel AG & Co. KGaA (DE) 2010-12-22 EP disclosed
WO-2010127902-A2 FOIL APPLICATOR HENKEL AG & CO. KGAA (DE) 2010-11-11 WO disclosed
WO-2010054981-A2 COMBINATION OF CATIONIC BLEACH ACTIVATORS AND DYES HENKEL AG & CO. KGAA (DE) 2010-05-20 WO disclosed
WO-2010015441-A1 MATTING ADDITIVE FOR BLOND HAIR DYING HENKEL AG & CO. KGAA (DE) 2010-02-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110162671-A1 BLEACHING AGENT COMPRISING 2-ACYLPYRIDINIUM DERIVATIVES KRT18, CBR3, ACOX3 CYP2D6 758/4885CYP2C19 1434/4885HSP90AA1 2500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.