SCHEMBL29059145

SCHEMBL29059145

CCc1c(C(=O)O)c2cc(OC)ccc2n1-c1ccc(C(C)(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.58
KMT2A Q03164 5/20 0.58
KDM4E B2RXH2 5/20 0.55
PPARG P37231 3/20 0.52
HTT P42858 3/20 0.48
MAPT P10636 2/20 0.48
HSD17B10 Q99714 2/20 0.47
PPARA Q07869 1/20 0.46
GAA P10253 1/20 0.45
PLA2G2A P14555 1/20 0.44
CCR9 P51686 1/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 3/20 0.42
PKM P14618 1/20 0.42
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HIF1A Q16665 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29059296 0.88 MEN1 (0.53) MEN1KMT2AKDM4EPPARGHTT
SCHEMBL29059277 0.85 KDM4E (0.76) MEN1KMT2AKDM4EPPARGHTT
SCHEMBL29059242 0.79 MEN1 (0.63) MEN1KMT2AKDM4EHTTMAPT
SCHEMBL29059297 0.79 NR1H4 (0.49) MEN1KMT2AKDM4EPPARGHTT
SCHEMBL29059180 0.79 MEN1 (0.52) MEN1KMT2AKDM4EHTTMAPT
SCHEMBL334350 0.76 PTGES (0.52) MEN1KMT2AKDM4EPPARGPPARA
SCHEMBL334428 0.75 AKR1C3 (0.50) MEN1KMT2AKDM4EPPARGHTT
SCHEMBL29059274 0.75 KMT2A (0.60) MEN1KMT2AKDM4EHTTMAPT
SCHEMBL1407523 0.74 PPARG (0.49) MEN1KMT2AKDM4EPPARGHTT
SCHEMBL29059391 0.74 MEN1 (0.56) MEN1KMT2AKDM4EPPARGHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116396205-B N-aryl indole derivative and preparation method and application thereof 沈阳药科大学 2024-10-01 CN disclosed
CN-116396205-A N-aryl indole derivative and preparation method and application thereof 沈阳药科大学 2023-07-07 CN disclosed