SCHEMBL29059153

SCHEMBL29059153

COc1cc2c(cc1OC)C(Cc1ccc(OC)c(OCc3ccccc3)c1)N(Cc1ccccc1)CC2

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.62
HCRTR2 O43614 9/20 0.62
LMNA P02545 2/20 0.59
KDM4E B2RXH2 1/20 0.59
ALDH1A1 P00352 1/20 0.59
MAPK1 P28482 1/20 0.59
HSD17B10 Q99714 1/20 0.59
CYP2D6 P10635 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11241355 0.90 HCRTR1 (0.60) HCRTR1HCRTR2LMNAKDM4EALDH1A1
SCHEMBL30585089 0.88 LMNA (0.79) LMNAKDM4EALDH1A1MAPK1HSD17B10
SCHEMBL9585990 0.88 LMNA (0.79) LMNAKDM4EALDH1A1MAPK1HSD17B10
SCHEMBL6382399 0.84 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL6381558 0.84 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL6380554 0.84 HCRTR1 (0.90) HCRTR1HCRTR2
SCHEMBL9416638 0.83 MTNR1B (0.67) HCRTR1HCRTR2LMNA
SCHEMBL6376398 0.81 HCRTR1 (0.72) HCRTR1HCRTR2
SCHEMBL3051846 0.80 CHRNA7 (0.54) HCRTR1HCRTR2
SCHEMBL6788304 0.80 HCRTR1 (0.88) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116655531-A Tetrandrine simplified substance for specifically inhibiting P-gp to reverse tumor multidrug resistance, and preparation method and application thereof 中国人民解放军陆军军医大学 2023-08-29 CN disclosed