SCHEMBL2905955

SCHEMBL2905955

N#Cc1cc2ccccc2nc1N[C@@H]1CCc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.45
EGFR P00533 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
KCNN3 Q9UGI6 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
FADS1 O60427 1/20 0.42
GLP1R P43220 1/20 0.42
PDPK1 O15530 1/20 0.41
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
PFKFB3 Q16875 1/20 0.40
CDK1 P06493 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
BCHE P06276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2906202 0.81 GBA1 (0.47) GBA1EGFRHDAC6KCNN3FADS1
SCHEMBL2904940 0.81 GBA1 (0.47) GBA1EGFRHDAC6KCNN3FADS1
SCHEMBL2906027 0.78 GBA1 (0.45) GBA1EGFRHDAC6KCNN3FADS1
SCHEMBL6071494 0.77 ACHE (0.50) KDM4EALDH1A1GAAKMT2ARXFP1
SCHEMBL2905886 0.76 PRKCQ (0.48) GBA1EGFRHDAC6KCNN3KDM4E
SCHEMBL2905882 0.76 PRKCQ (0.48) GBA1EGFRHDAC6KCNN3KDM4E
SCHEMBL2904936 0.76 AURKA (0.56) GBA1EGFRHDAC6KCNN3FADS1
SCHEMBL5117363 0.76 ACHE (0.49) KDM4EALDH1A1GAAKMT2ARXFP1
SCHEMBL1616604 0.74 GBA1 (0.43) GBA1EGFRHDAC6KCNN3FADS1
SCHEMBL3407222 0.74 LMNA (0.41) EGFRHDAC6KCNN3ALDH1A1FADS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP disclosed