SCHEMBL2905970

SCHEMBL2905970

Fc1ccc(Nc2cc3ccccc3nc2N[C@@H]2CCc3ccccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.44
CDK1 P06493 2/20 0.43
PFKFB3 Q16875 2/20 0.41
FADS1 O60427 1/20 0.41
EGFR P00533 1/20 0.41
PDPK1 O15530 1/20 0.40
MAPK14 Q16539 1/20 0.39
GLP1R P43220 1/20 0.39
MERTK Q12866 1/20 0.39
HDAC6 Q9UBN7 1/20 0.38
KCNN3 Q9UGI6 1/20 0.38
ROCK1 Q13464 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1615579 0.77 PFKFB3 (0.42) GBA1PFKFB3FADS1PDPK1MAPK14
SCHEMBL2904940 0.77 GBA1 (0.47) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2906202 0.77 GBA1 (0.47) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2905947 0.74 GLP1R (0.42) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2905955 0.74 GBA1 (0.45) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2906027 0.74 GBA1 (0.45) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2897916 0.73 GLP1R (0.49) GBA1PFKFB3GLP1RHDAC6KCNN3
SCHEMBL2905882 0.72 PRKCQ (0.48) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2905886 0.72 PRKCQ (0.48) GBA1CDK1PFKFB3FADS1EGFR
SCHEMBL2904936 0.72 AURKA (0.56) GBA1FADS1EGFRPDPK1GLP1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed