SCHEMBL29060147

SCHEMBL29060147

OC(O)(c1cc(Br)ccn1)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LOXL2 Q9Y4K0 2/20 0.34
RAD51 Q06609 1/20 0.34
SMARCA2 P51531 1/20 0.33
SMARCA4 P51532 1/20 0.33
LOX P28300 1/20 0.33
SYK P43405 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
SLC22A12 Q96S37 1/20 0.32
DGAT1 O75907 1/20 0.32
NT5E P21589 1/20 0.31
HSD11B1 P28845 1/20 0.31
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28400269 0.81 HSD11B1 (0.40) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL484767 0.79 LOXL2 (0.52) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL29581126 0.79 LOXL2 (0.52) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL28406030 0.78 SMN1; SMN2 (0.38) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL29620499 0.78 KDM4E (0.39) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL20875536 0.78 KDM4E (0.39) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
Bromide SCHEMBL15720464 0.78 LOXL2 (0.50) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
Ammonia Solution, Strong SCHEMBL27910510 0.78 LOXL2 (0.50) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL15801545 0.77 KDM4E (0.36) SMN1; SMN2KDM4EALDH1A1LOXL2RAD51
SCHEMBL3322613 0.76 SMN1; SMN2 (0.42) SMN1; SMN2KDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116670140-A Macrocyclic compounds containing 1,3, 4-oxadiazole rings as modulators of cystic fibrosis transmembrane conductance regulator 弗特克斯药品有限公司 2023-08-29 CN disclosed