SCHEMBL29065959

SCHEMBL29065959

O=Cc1cnc(-c2ccc(Br)cc2)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.48
HDAC3 O15379 4/20 0.42
HDAC4 P56524 4/20 0.42
HDAC1 Q13547 4/20 0.42
HDAC7 Q8WUI4 4/20 0.42
HDAC2 Q92769 4/20 0.42
HDAC10 Q969S8 4/20 0.42
HDAC11 Q96DB2 4/20 0.42
HDAC8 Q9BY41 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
HDAC9 Q9UKV0 4/20 0.42
HDAC5 Q9UQL6 4/20 0.42
IDO1 P14902 1/20 0.38
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA5A P35218 1/20 0.37
CA5B Q9Y2D0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16032766 0.82 HDAC1 (0.48) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1314645 0.82 PTPN11 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL850770 0.82 SMN1; SMN2 (0.51) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9394 0.81 ALDH1A1 (0.50) HDAC1HDAC6ALDH1A1KDM4EMAPT
SCHEMBL29183399 0.81 ALDH1A1 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL23146389 0.80 CDC7 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8336785 0.78 KMO (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL12151093 0.78 NPC1 (0.40) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL1849553 0.78 GAA (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL23146302 0.78 KDM4E (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116715639-A O-phenylenediamine and hydrazide-based targeting HDAC/PD-L1 bifunctional molecule synthesis and application thereof 南方医科大学 2023-09-08 CN disclosed