SCHEMBL29068379

SCHEMBL29068379

CC(F)(Oc1ccc(Br)cc1)C(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.41
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
MAPT P10636 2/20 0.33
LDHA P00338 1/20 0.33
WDR5 P61964 1/20 0.33
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP2A6 P11509 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PPARD Q03181 2/20 0.31
PPARA Q07869 2/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3945050 0.81 TRPV1 (0.51) TRPV1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL9926 0.80 ALDH1A1 (0.42) TRPV1ALDH1A1MAPTMAPK1RAB9A
SCHEMBL16546592 0.79 ALDH1A1 (0.40) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL28986637 0.76 ALDH1A1 (0.37) TRPV1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL23149109 0.75 ALDH1A1 (0.38) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL21078838 0.74 HSD17B10 (0.61) TRPV1ALDH1A1KMT2AMAPK1TSHR
SCHEMBL220074 0.73 MAPT (0.47) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL9243983 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL1006518 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL29217709 0.73 THRB (0.35) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111936503-B Oxazine monoacylglycerol lipase (MAGL) inhibitors 豪夫迈·罗氏有限公司 2023-09-12 CN disclosed