SCHEMBL290706

SCHEMBL290706

CC(C)(C)OC(=O)Nc1cnc(-c2cncc(F)c2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.39
DYRK1A Q13627 3/20 0.38
PIK3CG P48736 1/20 0.38
POLQ O75417 1/20 0.37
PRKACA P17612 1/20 0.37
ROCK1 Q13464 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
CYP17A1 P05093 3/20 0.36
CSNK2A2 P19784 1/20 0.36
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3744202 0.80 DYRK1A (0.43) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL19450126 0.80 NAMPT (0.51) PRKACAROCK1CYP17A1NAMPT
SCHEMBL13048243 0.79 DYRK1A (0.41) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL30617081 0.79 DYRK1A (0.41) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL13074537 0.79 DYRK1A (0.41) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL28254321 0.79 CSNK2A2 (0.47) PRKACAROCK1HDAC3HDAC4HDAC1
SCHEMBL289332 0.78 DYRK1A (0.42) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL13048201 0.78 DYRK1A (0.40) SYKDYRK1APIK3CGPOLQCYP17A1
SCHEMBL297950 0.76 CYP11B2 (0.33) DYRK1APIK3CGPOLQABL1RPS6KB1
SCHEMBL28184678 0.76 SYK (0.41) SYKNAMPTLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614826-B1 Process for preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2017-03-01 EP disclosed
US-9357780-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2016-06-07 US disclosed
EP-2427191-B1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2016-03-16 EP disclosed
EP-2614825-B1 Process for the preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2016-03-16 EP disclosed
EP-2604267-B1 Process for the preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2016-02-03 EP disclosed
EP-2604268-B1 Process for the preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2015-09-16 EP disclosed
US-9006446-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2015-04-14 US disclosed
US-20150045218-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2015-02-12 US disclosed
US-20140348947-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2014-11-27 US disclosed
US-8853246-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2014-10-07 US disclosed
EP-2614825-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-07-17 EP disclosed
EP-2604268-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-06-19 EP disclosed
EP-2604267-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-06-19 EP disclosed
US-20130089622-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-04-11 US disclosed
US-20130072382-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-03-21 US disclosed
US-8350044-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2013-01-08 US disclosed
EP-2427191-A1 PESTICIDAL COMPOSITIONS Dow AgroSciences LLC (US) 2012-03-14 EP disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed
WO-2010129497-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-11 WO disclosed
WO-2010129497-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100292253-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 SYK 3796/4885DYRK1A 3841/4885PIK3CG 795/4885
US-20130089622-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 SYK 3796/4885DYRK1A 3841/4885PIK3CG 795/4885
US-20140348947-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 SYK 3796/4885DYRK1A 3841/4885PIK3CG 795/4885
US-20150045218-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 SYK 3796/4885DYRK1A 3841/4885PIK3CG 795/4885
US-20130072382-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 SYK 3796/4885DYRK1A 3841/4885PIK3CG 795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.