SCHEMBL2908060

SCHEMBL2908060

COc1cc(F)ccc1OC1CCCC1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 10/20 0.51
RECQL P46063 1/20 0.50
PDE4B Q07343 8/20 0.48
PDE4D Q08499 8/20 0.48
PDE4C Q08493 6/20 0.48
POLB P06746 1/20 0.46
GLRA3 O75311 1/20 0.45
GLRB P48167 1/20 0.45
PDE3A Q14432 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19641654 0.97 PDE4A (0.48) PDE4ARECQLPDE4BPDE4DPDE4C
SCHEMBL5374046 0.85 SLC6A2 (0.54) PDE4B
SCHEMBL17210757 0.82 HTR2C (0.53) GLRA3GLRB
SCHEMBL14409244 0.81 OXTR (0.44) PDE4APDE4BPDE4DPDE4C
SCHEMBL2907378 0.81 ACHE (0.59) PDE4ARECQLPDE4BPDE4DPDE4C
SCHEMBL24925307 0.81 EIF4E (0.43) PDE4A
SCHEMBL24180131 0.80 PDE4A (0.44) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL5084709 0.80 CA12 (0.54) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL3457608 0.79 PDE4A (0.51) PDE4ARECQLPDE4BPDE4DPDE4C
SCHEMBL10196687 0.79 ACHE (0.57) PDE4ARECQLPDE4BPDE4DPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692109-B1 PHOSPHODIESTERASE 4 INHIBITORS, INCLUDING N-SUBSTITUTED DIARYLAMINE ANALOGS MEMORY PHARM CORP (US) 2010-08-18 EP disclosed
CN-1922144-A Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs MEMORY PHARM CORP (US) 2007-02-28 CN disclosed
EP-1692109-A2 PHOSPHODIESTERASE 4 INHIBITORS, INCLUDING N-SUBSTITUTED DIARYLAMINE ANALOGS Memory Pharmaceuticals Corporation (US) 2006-08-23 EP disclosed
US-20050222207-A1 Phosphodiesterase 4 inhibitors, including N-substituted diarylamine analogs MEMORY PHARMACEUTICAL CORPORATION 2005-10-06 US disclosed
WO-2005061458-A2 PHOSPHODIESTERASE 4 INHIBITORS, INCLUDING N-SUBSTITUTED DIARYLAMINE ANALOGS MEMORY PHARMACEUTICALS CORPORATION (US) 2005-07-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050222207-A1 Phosphodiesterase 4 inhibitors, including N-substituted diarylamine analogs PDE4A, PDE4B, PDE3B PDE4A 1/4885RECQL 137/4885PDE4B 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.