SCHEMBL29099495

SCHEMBL29099495

Cc1nc(N)sc1-c1ccc2c(c1)C(C(F)(F)F)CNC2=O

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 10/20 0.36
HRH1 P35367 10/20 0.36
HRH4 Q9H3N8 10/20 0.36
HRH3 Q9Y5N1 10/20 0.36
PI4KB Q9UBF8 1/20 0.33
JAK2 O60674 1/20 0.33
MKNK1 Q9BUB5 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
XBP1 P17861 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MPL P40238 1/20 0.31
CDC7 O00311 1/20 0.30
CDK9 P50750 1/20 0.30
ATAD2 Q6PL18 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29099527 0.84 HRH2 (0.37) HRH2HRH1HRH4HRH3PI4KB
SCHEMBL30185592 0.84 HRH2 (0.37) HRH2HRH1HRH4HRH3PI4KB
SCHEMBL29099575 0.74 PIK3CA (0.63) PI4KB
SCHEMBL29099574 0.74 PIK3CA (0.63) PI4KB
SCHEMBL30185577 0.74 PIK3CA (0.63) PI4KB
SCHEMBL31412980 0.73 PARP10 (0.44) MKNK1KDM4ELMNA
SCHEMBL29099501 0.70 HRH2 (0.35) HRH2HRH1HRH4HRH3PI4KB
SCHEMBL31544001 0.70 PRMT6 (0.37) HRH2HRH1HRH4HRH3JAK2
SCHEMBL30185591 0.69 HRH2 (0.36) HRH2HRH1HRH4HRH3JAK2
SCHEMBL29099535 0.69 HRH2 (0.36) HRH2HRH1HRH4HRH3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-B PI3K alpha inhibitor with double-ring structure, and preparation method and application thereof 生物岛实验室 2025-03-28 CN disclosed
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed