SCHEMBL29099501

SCHEMBL29099501

Cc1nc(N)sc1-c1ccc2c(c1)C(C(F)(F)F)C(=O)N=C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 9/20 0.35
HRH1 P35367 9/20 0.35
HRH4 Q9H3N8 9/20 0.35
HRH3 Q9Y5N1 9/20 0.35
GPR52 Q9Y2T5 5/20 0.32
PI4KB Q9UBF8 1/20 0.32
JAK2 O60674 1/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
XBP1 P17861 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
MPL P40238 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29099527 0.72 HRH2 (0.37) HRH2HRH1HRH4HRH3GPR52
SCHEMBL30185592 0.72 HRH2 (0.37) HRH2HRH1HRH4HRH3GPR52
SCHEMBL29099495 0.70 HRH2 (0.36) HRH2HRH1HRH4HRH3PI4KB
SCHEMBL31544001 0.66 PRMT6 (0.37) HRH2HRH1HRH4HRH3GPR52
SCHEMBL30185591 0.65 HRH2 (0.36) HRH2HRH1HRH4HRH3GPR52
SCHEMBL29099535 0.65 HRH2 (0.36) HRH2HRH1HRH4HRH3GPR52
SCHEMBL330359 0.64 BRD4 (0.51) HRH2HRH1HRH4HRH3GPR52
SCHEMBL48693 0.64 PIK3CD (0.65) HRH2HRH1HRH4HRH3GPR52
SCHEMBL330449 0.63 MAPT (0.53) HRH2HRH1HRH4HRH3KDM4E
SCHEMBL15801542 0.63 PIK3CA (0.51) PI4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed