SCHEMBL29099545

SCHEMBL29099545

O=C1CC(C(F)(F)F)c2cc(Br)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.43
AR P10275 2/20 0.39
ADRA2A P08913 1/20 0.37
PNMT P11086 1/20 0.37
S100A4 P26447 1/20 0.37
CYP1A2 P05177 1/20 0.36
MAPK1 P28482 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
KDM1A O60341 2/20 0.34
EDNRB P24530 1/20 0.34
EDNRA P25101 1/20 0.34
METAP1 P53582 2/20 0.33
PTPRC P08575 1/20 0.33
CYP19A1 P11511 1/20 0.33
TDP2 O95551 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP11 Q9NR21 1/20 0.33
BCL2 P10415 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30935380 1.00 PBRM1 (0.43) PBRM1ARADRA2APNMTS100A4
SCHEMBL26510292 0.78 PARP10 (0.44) ADRA2APNMTS100A4CYP1A2MAPK1
SCHEMBL4419838 0.74 PBRM1 (0.50) PBRM1ARADRA2APNMTS100A4
SCHEMBL2978084 0.72 LMNA (0.67) PBRM1ARLMNAGAAEDNRB
SCHEMBL30917500 0.71 CYP1A2 (0.41) PBRM1ARADRA2APNMTS100A4
SCHEMBL30917758 0.71 CYP1A2 (0.41) PBRM1ARADRA2APNMTS100A4
SCHEMBL30917876 0.71 CYP1A2 (0.41) PBRM1ARADRA2APNMTS100A4
SCHEMBL27864834 0.70 EDNRB (0.47) PBRM1ARS100A4EDNRBEDNRA
SCHEMBL30078429 0.69 MAOB (0.31) KDM1A
SCHEMBL16693108 0.68 DRD2 (0.41) ADRA2APNMTLMNAKDM1ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115611883-B PI3K alpha inhibitor with double-ring structure, and preparation method and application thereof 生物岛实验室 2025-03-28 CN disclosed
CN-115611883-A PI3K alpha inhibitor with bicyclic structure and preparation method and application thereof 生物岛实验室 2023-01-17 CN disclosed