SCHEMBL2910322

SCHEMBL2910322

C[C@@H](O)CNC(=O)c1cn(CCCNc2ccc([N+](=O)[O-])c(N)n2)cc1-c1ccc(C#N)cc1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.33
PRF1 P14222 1/20 0.33
EP300 Q09472 5/20 0.33
HAT1 O14929 3/20 0.33
GSK3B P49841 2/20 0.33
GSK3A P49840 1/20 0.33
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
MAP4K4 O95819 1/20 0.31
MINK1 Q8N4C8 1/20 0.31
TNIK Q9UKE5 1/20 0.31
NAMPT P43490 2/20 0.31
MAPK8 P45983 1/20 0.31
KAT2B Q92831 1/20 0.31
KDM1A O60341 1/20 0.30
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907197 1.00 SCN9A (0.33) SCN9APRF1EP300HAT1GSK3B
SCHEMBL2911588 0.91 ALDH1A1 (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2911036 0.91 ALDH1A1 (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2908179 0.90 MET (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2938731 0.90 MET (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2907242 0.90 LMNA (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2912251 0.90 SMN1; SMN2 (0.40) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2904193 0.90 SMN1; SMN2 (0.40) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2904632 0.90 LMNA (0.34) GSK3BGSK3AALDH1A1SMN1; SMN2
SCHEMBL2911391 0.90 GSK3B (0.33) GSK3BGSK3AALDH1A1SMN1; SMN2KAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed