SCHEMBL29109657

SCHEMBL29109657

Nc1ncc2ccccc2n1.c1cnc(-c2cnccn2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.46
CLK1 P49759 3/20 0.45
DYRK1A Q13627 2/20 0.45
CSNK1D P48730 1/20 0.45
CSNK1E P49674 1/20 0.45
ALOX5AP P20292 1/20 0.41
FEN1 P39748 1/20 0.41
LCK P06239 1/20 0.40
KDR P35968 1/20 0.40
JAK3 P52333 1/20 0.40
MAPK14 Q16539 1/20 0.40
DHFR P00374 1/20 0.40
DUSP4 Q13115 1/20 0.40
PTP4A1 Q93096 1/20 0.40
CYP3A4 P08684 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PI4KA P42356 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29509257 0.84 LCK (0.50) CLK1DYRK1ACSNK1DCSNK1ELCK
SCHEMBL41506 0.84 LCK (0.50) CLK1DYRK1ACSNK1DCSNK1ELCK
Hydrochloric Acid SCHEMBL29486326 0.82 LCK (0.49) CLK1DYRK1ACSNK1DCSNK1ELCK
Hydrochloric Acid SCHEMBL3468306 0.82 LCK (0.49) CLK1DYRK1ACSNK1DCSNK1ELCK
Hydrochloric Acid SCHEMBL28230152 0.82 LCK (0.49) CLK1DYRK1ACSNK1DCSNK1ELCK
Biphenyl SCHEMBL28889831 0.81 ADORA2A (0.51) CLK1DYRK1ACSNK1DCSNK1ELCK
Hydrochloric Acid SCHEMBL17237902 0.80 LCK (0.47) CLK1DYRK1ACSNK1DCSNK1ELCK
SCHEMBL28802825 0.79 CYP1A2 (0.54) METAP2DUSP4PTP4A1CYP3A4EGFR
SCHEMBL31418349 0.77 RAB9A (0.55) METAP2DUSP4PTP4A1CYP3A4CYP1A2
Quinoline SCHEMBL9745228 0.75 ALDH1A1 (0.65) METAP2DUSP4PTP4A1CYP3A4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115353507-B Biphenyl pyrazine quinazoline diamine, synthesis, activity and application thereof 首都医科大学 2023-10-20 CN disclosed