SCHEMBL2911026

SCHEMBL2911026

C[C@H](CO)NC(=O)c1cn(CCCNc2ccc(C(F)(F)F)cn2)cc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.40
FEN1 P39748 2/20 0.40
HCRTR1 O43613 4/20 0.40
CNR1 P21554 1/20 0.39
F10 P00742 1/20 0.38
PPARD Q03181 1/20 0.38
TACR1 P25103 2/20 0.36
TACR3 P29371 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
TRPV1 Q8NER1 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910207 1.00 ALOX5AP (0.40) ALOX5APFEN1HCRTR1CNR1F10
SCHEMBL2904248 0.88 PPARD (0.41) HCRTR1CNR1F10PPARDPRKAB2
SCHEMBL2904288 0.88 PPARD (0.41) HCRTR1CNR1F10PPARDPRKAB2
SCHEMBL2912436 0.86 F10 (0.41) HCRTR1CNR1F10PPARDPRKAB2
SCHEMBL2911030 0.86 GSK3B (0.46) ACVR1BTGFBR1ACVRL1ACVR1AHR
SCHEMBL2911764 0.86 GSK3B (0.46) ACVR1BTGFBR1ACVRL1ACVR1AHR
SCHEMBL2910724 0.85 GSK3B (0.42) KDM4EALDH1A1POLBAHR
SCHEMBL2912944 0.85 GSK3B (0.42) KDM4EALDH1A1POLBAHR
SCHEMBL2909829 0.83 HCRTR1 (0.41) HCRTR1CNR1F10PPARDTACR1
SCHEMBL2910831 0.78 GSK3B (0.48) ALDH1A1POLBAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed