SCHEMBL2912436

SCHEMBL2912436

O=C(O)c1cn(CCCNc2ccc(C(F)(F)F)cn2)cc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.41
PPARD Q03181 1/20 0.41
HCRTR1 O43613 4/20 0.40
GCGR P47871 5/20 0.39
GSK3B P49841 1/20 0.39
SORT1 Q99523 1/20 0.39
CNR1 P21554 1/20 0.39
PRKAB2 O43741 1/20 0.38
PRKAG1 P54619 1/20 0.38
PRKAA2 P54646 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAG3 Q9UGI9 1/20 0.38
PRKAG2 Q9UGJ0 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
CRHR1 P34998 1/20 0.38
RPS6KA3 P51812 1/20 0.38
HCRTR2 O43614 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2909829 0.88 HCRTR1 (0.41) F10PPARDHCRTR1GCGRCNR1
SCHEMBL2910207 0.86 ALOX5AP (0.40) F10PPARDHCRTR1GCGRCNR1
SCHEMBL2904248 0.86 PPARD (0.41) F10PPARDHCRTR1GCGRCNR1
SCHEMBL2904288 0.86 PPARD (0.41) F10PPARDHCRTR1GCGRCNR1
SCHEMBL2911026 0.86 ALOX5AP (0.40) F10PPARDHCRTR1GCGRCNR1
SCHEMBL2909840 0.84 GSK3B (0.55) GSK3B
SCHEMBL2912974 0.83 GSK3B (0.47) GSK3B
SCHEMBL1219415 0.75 GSK3B (0.51) GSK3B
SCHEMBL2913408 0.73 GSK3B (0.43) GSK3BCNR1
SCHEMBL3261753 0.73 ALDH1A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed