SCHEMBL2909829

SCHEMBL2909829

CC(C)(C)OC(=O)c1cn(CCCNc2ccc(C(F)(F)F)cn2)cc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 12/20 0.41
CNR1 P21554 2/20 0.39
F10 P00742 1/20 0.38
PPARD Q03181 1/20 0.38
HCRTR2 O43614 4/20 0.37
TACR1 P25103 2/20 0.36
TACR3 P29371 2/20 0.36
CNR2 P34972 1/20 0.36
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
GCGR P47871 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2912436 0.88 F10 (0.41) HCRTR1CNR1F10PPARDHCRTR2
SCHEMBL2913408 0.86 GSK3B (0.43) CNR1CNR2
SCHEMBL2904288 0.83 PPARD (0.41) HCRTR1CNR1F10PPARDHCRTR2
SCHEMBL2904248 0.83 PPARD (0.41) HCRTR1CNR1F10PPARDHCRTR2
SCHEMBL2910207 0.83 ALOX5AP (0.40) HCRTR1CNR1F10PPARDHCRTR2
SCHEMBL2911026 0.83 ALOX5AP (0.40) HCRTR1CNR1F10PPARDHCRTR2
SCHEMBL1219461 0.79 GSK3B (0.49) CNR1CNR2
SCHEMBL1219591 0.77 CNR1 (0.43) CNR1CNR2
SCHEMBL2909927 0.77 GSK3B (0.49) CNR1CNR2
SCHEMBL2909840 0.73 GSK3B (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537099-B1 PYRROLE BASED INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 NOVARTIS VACCINES & DIAGNOSTIC (US) 2010-08-11 EP disclosed