SCHEMBL29120691

SCHEMBL29120691

COc1c(Nc2ccc3ncccc3c2)c(=O)c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.54
STK10 O94804 1/20 0.52
SLK Q9H2G2 1/20 0.52
NPC1 O15118 4/20 0.50
RAB9A P51151 3/20 0.50
MAPT P10636 2/20 0.49
POLB P06746 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
HTT P42858 2/20 0.47
ALOX15 P16050 1/20 0.47
NOTUM Q6P988 1/20 0.46
JAK2 O60674 1/20 0.45
JAK3 P52333 1/20 0.45
PTK2 Q05397 1/20 0.45
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
BRAF P15056 1/20 0.44
GRM4 Q14833 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29120695 0.86 NPC1 (0.61) IGF1RSTK10SLKNPC1RAB9A
SCHEMBL8674402 0.82 NPC1 (0.52) STK10SLKNPC1RAB9AMAPT
SCHEMBL29120686 0.81 ALDH1A1 (0.59) STK10SLKNPC1RAB9AMAPT
SCHEMBL8668406 0.80 NPC1 (0.52) STK10SLKNPC1RAB9AMAPT
SCHEMBL7354053 0.79 PLK1 (0.50) STK10SLKNPC1RAB9AMAPT
SCHEMBL29120687 0.79 ALDH1A1 (0.53) STK10SLKNPC1RAB9AMAPT
SCHEMBL28243562 0.76 NPC1 (0.66) IGF1RSTK10SLKNPC1RAB9A
SCHEMBL29120689 0.76 BRAF (0.47) STK10SLKNPC1RAB9AMAPT
SCHEMBL29120693 0.75 SYK (0.54) STK10SLKNPC1MAPTPOLB
SCHEMBL8669622 0.75 PLK1 (0.61) SLKAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116947756-B Cyclobutene diketo quinoline compound and preparation method, pharmaceutical composition and application thereof 中国药科大学 2025-02-07 CN disclosed
WO-2025025472-A1 CYCLOBUTENEDIONE-BASED QUINOLINE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 中国药科大学 2025-02-06 WO disclosed
CN-116947756-A Cyclobutene diketo quinoline compound and preparation method, pharmaceutical composition and application thereof 中国药科大学 2023-10-27 CN disclosed