SCHEMBL29124530

SCHEMBL29124530

COc1ccc(-n2cnn(CCBr)c2=O)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.49
BRD9 Q9H8M2 3/20 0.46
MCHR1 Q99705 3/20 0.43
HSD17B3 P37058 1/20 0.43
CYP2C9 P11712 1/20 0.40
CYP1A2 P05177 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29124533 0.85 ROCK2 (0.43) ROCK2HSD17B3L3MBTL1GAA
SCHEMBL29124531 0.82 HSD17B3 (0.57) ROCK2HSD17B3CYP2C9CYP1A2MAPT
SCHEMBL29124532 0.77 PPARD (0.46) ROCK2HSD17B3
SCHEMBL29124525 0.77 SMN1; SMN2 (0.44) ROCK2HSD17B3LMNA
SCHEMBL29124535 0.75 PPARD (0.44) ROCK2HSD17B3
SCHEMBL29124529 0.75 PPARD (0.44) ROCK2HSD17B3MAPT
SCHEMBL29124527 0.74 ALDH1A1 (0.45) ROCK2HSD17B3
SCHEMBL16196788 0.69 PPARD (0.47) ROCK2HSD17B3MAPT
SCHEMBL7458461 0.68 MAPT (0.56) HSD17B3GAAMAPTLMNA
SCHEMBL2393523 0.68 BRD9 (0.43) BRD9MCHR1CYP2C9CYP1A2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181156-B Hederagenin derivative and application thereof in preparation of antitumor drugs 延边大学 2023-11-10 CN disclosed