SCHEMBL29124533

SCHEMBL29124533

COc1cc(-n2cnn(CCBr)c2=O)cc(OC)c1OC

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B3 P37058 1/20 0.39
GAA P10253 1/20 0.38
CYP19A1 P11511 1/20 0.38
NQO2 P16083 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29124530 0.85 ROCK2 (0.49) ROCK2L3MBTL1HSD17B3GAA
SCHEMBL29124531 0.78 HSD17B3 (0.57) ROCK2KMT2AHSD17B3
SCHEMBL29124532 0.73 PPARD (0.46) ROCK2MEN1KMT2AHSD17B3
SCHEMBL29124527 0.72 ALDH1A1 (0.45) ROCK2HSD17B3
SCHEMBL29124529 0.70 PPARD (0.44) ROCK2HSD17B3
SCHEMBL29124535 0.70 PPARD (0.44) ROCK2HSD17B3
SCHEMBL29124525 0.69 SMN1; SMN2 (0.44) ROCK2HSD17B3
SCHEMBL3535318 0.64 HTR1A (0.44) ROCK2HSD17B3
SCHEMBL15033478 0.62 G6PD (0.61) MEN1KMT2AL3MBTL1GAA
SCHEMBL10975563 0.62 RAB9A (0.55) MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181156-B Hederagenin derivative and application thereof in preparation of antitumor drugs 延边大学 2023-11-10 CN disclosed