SCHEMBL29131028

SCHEMBL29131028

COc1cc(N2CCCS2(=O)=O)ccc1Br

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.48
TP53 P04637 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA6 P23280 1/20 0.43
OPRK1 P41145 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
POLB P06746 2/20 0.43
LMNA P02545 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 2/20 0.43
PDE4A P27815 1/20 0.43
P2RX7 Q99572 2/20 0.42
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31038304 0.80 TP53 (0.54) CHEK1TP53SMN1; SMN2POLBLMNA
SCHEMBL25229814 0.80 TP53 (0.54) CHEK1TP53SMN1; SMN2POLBLMNA
SCHEMBL14686719 0.80 TP53 (0.51) CHEK1TP53SMN1; SMN2POLBLMNA
SCHEMBL31079461 0.76 POLB (0.55) TP53SMN1; SMN2CA1CA2CA6
SCHEMBL25424710 0.76 POLB (0.55) TP53SMN1; SMN2CA1CA2CA6
SCHEMBL12445262 0.75 LMNA (0.60) TP53CA1CA2CA6OPRK1
SCHEMBL12445151 0.75 CA1 (0.47) TP53CA1CA2CA6OPRK1
SCHEMBL23705839 0.73 ALDH1A1 (0.55) SMN1; SMN2LMNA
SCHEMBL31091978 0.73 ALDH1A1 (0.55) SMN1; SMN2LMNA
SCHEMBL2360208 0.73 TP53 (0.45) CHEK1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117069724-A Fused ring compounds, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-17 CN disclosed