SCHEMBL29131069

SCHEMBL29131069

NC(=O)Oc1cccc(-c2ccnc(Cl)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
KMO O15229 3/20 0.46
KDM4E B2RXH2 3/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
DYRK1A Q13627 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
MAPT P10636 2/20 0.40
ESR1 P03372 1/20 0.40
HTT P42858 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
NFKB1 P19838 1/20 0.39
STAT3 P40763 1/20 0.39
STAT1 P42224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28669409 0.83 MAP4K4 (0.48) MEN1KMT2AKMOKDM4ENPC1
SCHEMBL29623827 0.83 MAP4K4 (0.48) MEN1KMT2AKMOKDM4ENPC1
SCHEMBL3397244 0.81 MAP4K4 (0.52) MEN1KMT2AKMOKDM4EDYRK1A
SCHEMBL14638214 0.79 DYRK1A (0.60) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL1469470 0.76 MAP4K4 (0.48) MEN1KMT2AKMOKDM4EDYRK1A
SCHEMBL823888 0.76 KMO (0.58) KMOKDM4ENPC1RAB9A
SCHEMBL14637950 0.75 GRM5 (0.49) MEN1KMT2AKMODYRK1ACLK4
SCHEMBL3401551 0.74 KMO (0.50) MEN1KMT2AKMOCLK4MAPT
SCHEMBL4326155 0.73 KMT2A (0.54) MEN1KMT2AKDM4ENPC1RAB9A
SCHEMBL823885 0.73 HSD17B1 (0.55) KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088851-A Pyrimidine amine NUAK inhibitor and preparation method and application thereof 特科罗生物科技(成都)有限公司 2023-11-21 CN disclosed