SCHEMBL29131925

SCHEMBL29131925

Oc1ccc(-c2ccnnc2)c(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.48
HSD17B2 P37059 1/20 0.48
WNT3A P56704 4/20 0.42
ESR2 Q92731 1/20 0.41
AR P10275 2/20 0.40
KIF11 P52732 1/20 0.38
PDE3B Q13370 2/20 0.37
PDE3A Q14432 2/20 0.37
S1PR1 P21453 2/20 0.36
TNIK Q9UKE5 1/20 0.36
ADH5 P11766 1/20 0.36
PDK1 Q15118 2/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
TRPA1 O75762 1/20 0.35
S1PR3 Q99500 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29276031 0.81 S1PR1 (0.35) HSD17B1HSD17B2WNT3AESR2KIF11
SCHEMBL14832293 0.79 CYP11B1 (0.56) HSD17B1HSD17B2PDE3BPDE3AS1PR1
SCHEMBL28415938 0.78 HSD17B1 (0.59) HSD17B1HSD17B2ESR2ARKIF11
SCHEMBL5792355 0.78 GLA (0.54) HSD17B1HSD17B2ESR2ARKIF11
SCHEMBL31256038 0.78 GLA (0.54) HSD17B1HSD17B2ESR2ARKIF11
SCHEMBL319582 0.75 SCN9A (0.41) WNT3AKIF11S1PR1
SCHEMBL321081 0.75 SCN9A (0.41) WNT3AKIF11S1PR1
SCHEMBL1802128 0.75 ALOX5 (0.59) HSD17B1HSD17B2ESR2ARKIF11
SCHEMBL29131926 0.75 ALOX5AP (0.50) KIF11S1PR1
SCHEMBL27870662 0.74 HSD17B1 (0.55) HSD17B1HSD17B2ESR2ARKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116969920-A Fused pyridazine derivative, preparation method and medical application thereof 上海辉启生物医药科技有限公司 2023-10-31 CN disclosed