SCHEMBL29132992

SCHEMBL29132992

COc1cc(-n2ccccc2=O)ccc1Br

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
F10 P00742 9/20 0.42
MAPT P10636 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
GRM4 Q14833 1/20 0.37
KLKB1 P03952 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529067 0.85 CYP1A2 (0.60) CYP1A2L3MBTL1F10MAPTCYP2C9
SCHEMBL8160058 0.81 CYP1A2 (0.46) CYP1A2L3MBTL1F10MAPTCYP3A4
SCHEMBL8148718 0.81 CYP1A2 (0.43) CYP1A2L3MBTL1F10MAPTCYP3A4
SCHEMBL6535853 0.79 CYP1A2 (0.47) CYP1A2L3MBTL1F10MAPTCYP3A4
SCHEMBL12545383 0.79 CYP1A2 (0.43) CYP1A2L3MBTL1F10MAPTCYP3A4
SCHEMBL28328775 0.78 ALDH1A1 (0.49) CYP1A2L3MBTL1F10
SCHEMBL8149820 0.78 PDE5A (0.46) CYP1A2L3MBTL1F10MAPTCYP3A4
SCHEMBL8164439 0.77 ALDH1A1 (0.57) CYP1A2L3MBTL1F10MAPT
SCHEMBL16296617 0.76 BIRC5 (0.47) CYP1A2L3MBTL1MAPT
SCHEMBL5097812 0.76 F10 (0.40) F10KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed