SCHEMBL29133079

SCHEMBL29133079

COCc1cc(C(=O)N(N)C(C)=O)ccc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCE Q02156 2/20 0.36
HPGD P15428 1/20 0.35
KMT2A Q03164 6/20 0.34
ALDH1A1 P00352 6/20 0.34
MEN1 O00255 5/20 0.34
MAPT P10636 5/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.34
HSP90AA1 P07900 2/20 0.33
HSP90AB1 P08238 2/20 0.33
CYP1A2 P05177 2/20 0.33
PARP10 Q53GL7 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 2/20 0.33
POLB P06746 1/20 0.33
PKM P14618 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30602390 0.82 ALDH1A1 (0.42) HPGDKMT2AALDH1A1MEN1HTT
SCHEMBL24595665 0.81 ALDH1A1 (0.48) HPGDKMT2AALDH1A1MEN1MAPT
SCHEMBL30622253 0.81 ALDH1A1 (0.48) HPGDKMT2AALDH1A1MEN1MAPT
SCHEMBL256775 0.80 MLYCD (0.41) HPGDKMT2AALDH1A1MEN1MAPT
SCHEMBL408849 0.77 CA1 (0.44) PRKCEALDH1A1HTTRAB9APOLB
SCHEMBL29133089 0.77 ALDH1A1 (0.53) KMT2AALDH1A1MEN1MAPTHTT
SCHEMBL256771 0.76 NOTUM (0.50) HPGDKMT2AALDH1A1MEN1MAPT
SCHEMBL30622268 0.76 NOTUM (0.50) HPGDKMT2AALDH1A1MEN1MAPT
SCHEMBL29133180 0.75 GSK3B (0.49) KMT2AALDH1A1MEN1MAPTGAA
SCHEMBL29133080 0.74 TP53 (0.41) KMT2AALDH1A1MEN1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed