SCHEMBL2913360

SCHEMBL2913360

CCc1nc2cc(OC)c(N3CCN(C)CC3)cc2c(Nc2ccccc2F)c1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 9/20 0.52
CSF1R P07333 9/20 0.52
KCNH2 Q12809 9/20 0.49
HTR1A P08908 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR2C P28335 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2911894 0.90 SCN5A (0.65) SCN5ACSF1RKCNH2
SCHEMBL2909682 0.85 CSF1R (0.64) SCN5ACSF1RKCNH2
SCHEMBL2909211 0.83 CSF1R (0.51) SCN5ACSF1RKCNH2
SCHEMBL2913426 0.81 CSF1R (0.51) SCN5ACSF1RKCNH2
SCHEMBL2911555 0.81 KCNH2 (0.53) SCN5ACSF1RKCNH2
SCHEMBL2912641 0.79 CSF1R (0.60) SCN5ACSF1RKCNH2HTR1AHTR1D
SCHEMBL2914061 0.79 CSF1R (0.49) SCN5ACSF1RKCNH2HTR1AHTR1D
SCHEMBL2913359 0.78 CSF1R (0.66) SCN5ACSF1RKCNH2
SCHEMBL2908767 0.77 CSF1R (0.83) SCN5ACSF1RKCNH2
SCHEMBL2911700 0.76 KCNH2 (0.51) SCN5ACSF1RKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed