SCHEMBL29133695

SCHEMBL29133695

CC1(C)OB(c2ccc3ncnc(NCCc4ccccc4)c3c2)OC1(C)C

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 7/20 0.57
EGFR P00533 4/20 0.57
MAPK1 P28482 2/20 0.57
LMNA P02545 2/20 0.57
APP P05067 2/20 0.57
CCNC P24863 1/20 0.56
CDKN1A P38936 1/20 0.56
CDK8 P49336 1/20 0.56
CDK19 Q9BWU1 1/20 0.56
CNR1 P21554 1/20 0.53
CNR2 P34972 1/20 0.53
PIK3CD O00329 1/20 0.52
PIK3R1 P27986 1/20 0.52
FYN P06241 1/20 0.50
SRC P12931 1/20 0.50
DYRK1A Q13627 1/20 0.48
NR2F2 P24468 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
SLC29A1 Q99808 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133792 0.78 PDPK1 (0.42) EGFRCCNCCDKN1ACDK8CDK19
SCHEMBL24576519 0.77 GALR3 (0.58) EGFRLMNADYRK1ANR2F2
SCHEMBL29775101 0.77 GALR3 (0.58) EGFRLMNADYRK1ANR2F2
SCHEMBL24576525 0.77 GALR3 (0.58) EGFRLMNADYRK1ANR2F2
SCHEMBL24609450 0.77 LMNA (0.56) EGFRLMNADYRK1ANR2F2
SCHEMBL13283269 0.76 HTT (0.76) HTTEGFRMAPK1LMNAAPP
SCHEMBL4741967 0.75 HTT (0.70) HTTEGFRMAPK1LMNAAPP
SCHEMBL9921509 0.75 PIK3CD (0.85) HTTEGFRMAPK1LMNAAPP
SCHEMBL13912334 0.75 EGFR (0.76) HTTEGFRMAPK1LMNAAPP
SCHEMBL13192080 0.75 HTT (0.70) HTTEGFRMAPK1LMNAAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117295716-A Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors 麦克尼斯迪克治疗有限公司 2023-12-26 CN disclosed