SCHEMBL29134476

SCHEMBL29134476

NC(=O)c1cccc(-c2ccncn2)c1-c1ccncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
BCAT2 O15382 1/20 0.42
JAK2 O60674 1/20 0.42
PARP1 P09874 2/20 0.41
CYP46A1 Q9Y6A2 2/20 0.41
CSNK1A1 P48729 1/20 0.41
TYRO3 Q06418 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
GRM5 P41594 1/20 0.41
AURKA O14965 1/20 0.39
PDK2 Q15119 1/20 0.38
CDC7 O00311 1/20 0.38
ADORA2B P29275 1/20 0.37
PLK4 O00444 1/20 0.37
MAPK13 O15264 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25421476 0.90 BCAT2 (0.51) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL16654579 0.87 BCAT2 (0.53) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL7098623 0.86 IKBKB (0.43) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL31329756 0.85 CHRNB2 (0.41) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL7098629 0.84 PARP1 (0.42) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL30692651 0.84 BCAT2 (0.50) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL21381430 0.81 JAK2 (0.41) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL21629952 0.81 SYK (0.39) CHRNB2CHRNB4CHRNA3CHRNA4BCAT2
SCHEMBL30882864 0.81 JAK2 (0.41) KEAP1NFE2L2CHRNB2CHRNB4CHRNA3
SCHEMBL21381429 0.80 JAK2 (0.41) KEAP1NFE2L2JAK2PARP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed