Thiophene Carboxylic Acid

Thiophene Carboxylic Acid

SCHEMBL29135074

NC(=O)c1cccc(S(=O)(=O)N2CCCc3ccccc32)c1.O=C(O)c1cccs1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.70
AKR1C1 Q04828 1/20 0.62
GAA P10253 1/20 0.59
MEN1 O00255 4/20 0.56
KMT2A Q03164 4/20 0.56
NR3C1 P04150 4/20 0.53
AR P10275 4/20 0.53
LMNA P02545 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
HTT P42858 2/20 0.53
STAT3 P40763 1/20 0.53
CASP3 P42574 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
ATM Q13315 1/20 0.53
TSHR P16473 1/20 0.52
KDM4E B2RXH2 2/20 0.51
MAPT P10636 2/20 0.51
HPGD P15428 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiophene Carboxylic Acid SCHEMBL29135071 0.89 KMT2A (0.69) AKR1C3MEN1KMT2ANR3C1LMNA
Benzoic Acid SCHEMBL29134718 0.89 AKR1C3 (0.84) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL29135079 0.86 AKR1C3 (0.72) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL29134731 0.85 GAA (0.61) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL30679105 0.84 AKR1C3 (1.00) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL664241 0.84 AKR1C3 (1.00) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL29135072 0.83 AKR1C3 (0.74) AKR1C3AKR1C1GAAMEN1KMT2A
SCHEMBL29134720 0.81 NR3C1 (0.61) AKR1C3AKR1C1GAANR3C1AR
SCHEMBL29134721 0.81 AKR1C3 (0.70) AKR1C3AKR1C1GAAMEN1KMT2A
2-Picolinic Acid SCHEMBL29135065 0.81 AKR1C3 (0.70) AKR1C3AKR1C1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117298108-A Androgen receptor and glucocorticoid receptor dual-target inhibitor and application thereof 浙江师范大学 2023-12-29 CN disclosed