SCHEMBL29136045

SCHEMBL29136045

O=C(O)c1cccc(Cn2cc(I)c3cc(Br)ccc3c2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 4/20 0.46
KMT2A Q03164 3/20 0.43
MRGPRX4 Q96LA9 2/20 0.43
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HIF1A Q16665 1/20 0.41
IDO1 P14902 1/20 0.41
POLB P06746 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 2/20 0.40
MEN1 O00255 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
P2RY2 P41231 1/20 0.39
FOLH1 Q04609 1/20 0.39
HPGD P15428 1/20 0.38
MEP1B Q16820 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30656595 1.00 MAPK8 (0.46) MAPK8KMT2AMRGPRX4CYP2D6CYP2C9
SCHEMBL29778984 0.87 BRD4 (0.47) MAPK8KMT2AMEN1SMN1; SMN2HPGD
SCHEMBL29778993 0.87 MAPK8 (0.59) MAPK8HIF1AIDO1ALDH1A1
SCHEMBL29136046 0.87 BRD4 (0.47) MAPK8KMT2AMEN1SMN1; SMN2HPGD
SCHEMBL29136019 0.79 KMT2A (0.45) MAPK8KMT2AMRGPRX4CYP2D6CYP2C9
SCHEMBL30656512 0.79 KMT2A (0.45) MAPK8KMT2AMRGPRX4CYP2D6CYP2C9
SCHEMBL30656549 0.77 IDO1 (0.51) MRGPRX4IDO1SMN1; SMN2
SCHEMBL29136018 0.77 IDO1 (0.51) MRGPRX4IDO1SMN1; SMN2
SCHEMBL2419642 0.77 LMNA (0.52) MAPK8KMT2AHTTMEN1SMN1; SMN2
SCHEMBL2420795 0.71 ALDH1A1 (0.48) MAPK8KMT2AIDO1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117136186-A Selective inhibitors of ROCK1 and ROCK2 protein kinases and uses thereof 盖诺斯克公司 2023-11-28 CN disclosed