SCHEMBL2913622

SCHEMBL2913622

CCOC(=O)c1cnc2cc(OC)c(Br)cc2c1Nc1ccc(F)cc1Cl

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 10/20 0.66
MAPT P10636 3/20 0.65
GAA P10253 1/20 0.65
THRB P10828 1/20 0.65
SRC P12931 1/20 0.51
CA2 P00918 1/20 0.49
NUDT1 P36639 3/20 0.49
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
PDE6D O43924 1/20 0.47
PDE5A O76074 1/20 0.47
PDE6A P16499 1/20 0.47
PDE6G P18545 1/20 0.47
PDE6B P35913 1/20 0.47
PDE6C P51160 1/20 0.47
PDE6H Q13956 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2913852 0.94 CSF1R (0.59) CSF1RMAPTGAATHRBSRC
SCHEMBL2905486 0.91 MAPT (0.67) CSF1RMAPTGAATHRBSRC
SCHEMBL2907950 0.91 CSF1R (0.65) CSF1RMAPTGAATHRBNUDT1
SCHEMBL2911260 0.89 CSF1R (0.65) CSF1RMAPTGAATHRBNUDT1
SCHEMBL2911338 0.88 MAPT (0.56) CSF1RMAPTGAATHRBLMNA
SCHEMBL2911733 0.88 CSF1R (0.66) CSF1RMAPTGAATHRBCA2
SCHEMBL2910481 0.88 CSF1R (0.65) CSF1RMAPTGAATHRBNUDT1
SCHEMBL2911907 0.86 CSF1R (0.66) CSF1RMAPTGAATHRBNUDT1
SCHEMBL2909819 0.86 MAPT (0.72) CSF1RMAPTGAATHRBSRC
SCHEMBL2913881 0.86 CSF1R (0.65) CSF1RMAPTGAATHRBSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010496-B1 4-ANILINOQUINOLINE-3-CARBOXAMIDES AS CSF-1R KINASE INHIBITORS ASTRAZENECA AB (SE) 2010-08-25 EP disclosed