SCHEMBL29136349

SCHEMBL29136349

Brc1cc(OCC2CCOCC2)cc(Br)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.40
DCPS Q96C86 1/20 0.40
XDH P47989 2/20 0.38
GRM5 P41594 3/20 0.37
ATXN2 Q99700 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
HTR3A P46098 1/20 0.36
KCNH2 Q12809 1/20 0.36
PIM1 P11309 1/20 0.35
CYP11B2 P19099 1/20 0.35
P2RX3 P56373 1/20 0.35
P2RX2 Q9UBL9 1/20 0.35
ACACB O00763 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
SLC2A1 P11166 1/20 0.35
MCHR1 Q99705 1/20 0.35
GRM4 Q14833 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29136326 0.86 DHFR (0.34) DHFRDCPSXDHGRM5CYP2D6
SCHEMBL29136313 0.83 GRM5 (0.41) XDHGRM5SLC6A2SLC6A4HTR3A
SCHEMBL20424133 0.79 LMNA (0.42) GRM5CYP2D6P2RX3P2RX2ACACB
SCHEMBL3103772 0.76 CHRNB2 (0.52) CYP2D6CYP11B2
SCHEMBL18481622 0.76 LMNA (0.45) GRM5CYP2D6SLC6A2P2RX3P2RX2
SCHEMBL20870755 0.76 TSHR (0.45) XDHACACB
SCHEMBL13096931 0.76 CYP2D6 (0.39) XDHATXN2CYP2D6CYP11B2P2RX3
SCHEMBL18471240 0.75 CYP2D6 (0.44) GRM5CYP2D6P2RX3P2RX2ACACB
SCHEMBL16031257 0.74 CYP2D6 (0.46) DHFRDCPSCYP2D6SLC2A1
SCHEMBL29136297 0.74 GRM5 (0.40) DHFRGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117343056-A Pyridopyrrole derivatives and their use in medicine 广东东阳光药业股份有限公司 2024-01-05 CN disclosed