SCHEMBL29136780

SCHEMBL29136780

C=CC(=O)Oc1cc(OC)ccc1Br

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
THRB P10828 2/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 1/20 0.42
POLB P06746 1/20 0.41
TGM2 P21980 1/20 0.41
NPC1 O15118 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27850566 0.84 CA12 (0.55) ALDH1A1THRBMEN1KMT2AMAPT
SCHEMBL6767178 0.83 ERN1 (0.47) ALDH1A1THRBMEN1KMT2AMAPT
SCHEMBL4269240 0.81 ALDH1A1 (0.44) ALDH1A1THRBMEN1KMT2AMAPT
SCHEMBL30406222 0.81 ALDH1A1 (0.53) ALDH1A1THRBMEN1KMT2AMAPT
SCHEMBL22381406 0.81 THRB (0.45) ALDH1A1THRBMAPTTGM2ABCG2
SCHEMBL6173663 0.80 BACE1 (0.56) ALDH1A1MEN1KMT2AMAPTPOLB
SCHEMBL27616513 0.80 PTGS1 (0.50) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL18869352 0.80 KDM4E (0.55) ALDH1A1THRBMEN1KMT2AMAPT
SCHEMBL28783574 0.78 TSHR (0.43) ALDH1A1ABCG2NFKB1
SCHEMBL10499949 0.78 KMT2A (0.44) ALDH1A1THRBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed