SCHEMBL29137007

SCHEMBL29137007

O=C(O)Cc1cn2cc(C3CC3)cc(Br)c2n1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
EPHX2 P34913 1/20 0.38
KLKB1 P03952 3/20 0.33
THRA P10827 2/20 0.33
THRB P10828 2/20 0.33
METTL3 Q86U44 1/20 0.32
PPARA Q07869 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27029949 0.85 KLKB1 (0.39) KDM4EALDH1A1EPHX2KLKB1METTL3
SCHEMBL24737489 0.83 PIK3R1 (0.33) EPHX2KLKB1
SCHEMBL24739338 0.83 KDM4E (0.38) KDM4EALDH1A1POLBTDP1THRB
SCHEMBL24739861 0.82 DRD2 (0.32)
SCHEMBL29136933 0.81 GRM5 (0.31) ALDH1A1EPHX2KLKB1METTL3RXFP1
SCHEMBL31658609 0.81 DRD2 (0.34)
SCHEMBL21355494 0.81 DRD2 (0.32) KLKB1
SCHEMBL21368003 0.81 DRD2 (0.32)
SCHEMBL24737556 0.80 RXFP1 (0.50) KDM4EALDH1A1TDP1L3MBTL1EPHX2
SCHEMBL24740076 0.79 HCAR3 (0.34) EPHX2KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed