SCHEMBL29137030

SCHEMBL29137030

NC(=O)OCc1cn2cc(C3CC3)cc(CCl)c2n1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.32
KLKB1 P03952 3/20 0.32
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27033928 0.90 KLKB1 (0.33) GRM5KLKB1MAPT
SCHEMBL29136933 0.83 GRM5 (0.31) GRM5KLKB1
SCHEMBL29137027 0.81 KLKB1 (0.33) GRM5KLKB1
SCHEMBL27033666 0.79 GRM5 (0.33) GRM5KLKB1
SCHEMBL24737346 0.76 CA1 (0.39) KLKB1
SCHEMBL21355124 0.76 SUV39H2 (0.32) KLKB1
SCHEMBL21355696 0.75 CYP4F2 (0.35) KLKB1MAPT
SCHEMBL27033822 0.75 KDM4E (0.33) GRM5KLKB1MAPT
SCHEMBL29137034 0.74 METTL3 (0.47) KLKB1
SCHEMBL21355085 0.74 KLKB1 (0.47) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed