SCHEMBL29139935

SCHEMBL29139935

CN(C)CCC(=O)N1CCC(c2ccccc2[C@H]2CCCN2c2ccc(Br)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.44
TMEM97 Q5BJF2 1/20 0.44
NAMPT P43490 1/20 0.39
BCL2 P10415 1/20 0.38
BCL2L1 Q07817 1/20 0.38
CYP2D6 P10635 3/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
SSTR1 P30872 4/20 0.36
SSTR3 P32745 4/20 0.36
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29139938 1.00 SIGMAR1 (0.44) SIGMAR1TMEM97NAMPTBCL2BCL2L1
SCHEMBL29855777 1.00 SIGMAR1 (0.44) SIGMAR1TMEM97NAMPTBCL2BCL2L1
SCHEMBL28532862 0.83 MAPT (0.41) CYP2D6ALDH1A1CYP1A2CYP3A4GAA
SCHEMBL29855898 0.82 MAPT (0.36) SIGMAR1TMEM97BCL2BCL2L1CYP2D6
SCHEMBL28522991 0.82 RBP4 (0.41) CYP2D6ALDH1A1CYP1A2CYP3A4GAA
SCHEMBL28527478 0.80 GPR119 (0.47) NAMPTMAPT
SCHEMBL28528284 0.79 CYP2D6 (0.38) CYP2D6CYP2C9CYP2C19HRH3
SCHEMBL28528279 0.79 CYP2D6 (0.38) CYP2D6CYP2C9CYP2C19HRH3
SCHEMBL28909558 0.78 HRH3 (0.41) CYP2D6MAPTCYP2C9CYP2C19HRH3
SCHEMBL28909552 0.78 HRH3 (0.41) CYP2D6MAPTCYP2C9CYP2C19HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed