SCHEMBL29140551

SCHEMBL29140551

Oc1ccc(Br)c(O)c1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
PDE4B Q07343 4/20 0.41
PDE4A P27815 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
ALOX5 P09917 1/20 0.40
ESR2 Q92731 2/20 0.40
ESR1 P03372 1/20 0.40
BACE1 P56817 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
AKR1C4 P17516 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29587494 1.00 CRHBP (0.48) CRHBPCRHR2PDE4BPDE4APDE4C
SCHEMBL8157958 0.84 CRHBP (0.45) CRHBPCRHR2PDE4BPDE4APDE4C
SCHEMBL7112114 0.83 CRHBP (0.43) CRHBPCRHR2ALOX5ESR2ESR1
SCHEMBL9348187 0.81 ALOX5 (0.46) PDE4BPDE4APDE4CPDE4DALOX5
SCHEMBL31275930 0.81 ALOX5 (0.46) PDE4BPDE4APDE4CPDE4DALOX5
SCHEMBL22891448 0.81 CRHBP (0.47) CRHBPCRHR2PDE4BPDE4APDE4C
SCHEMBL22891656 0.79 ESR2 (0.42) CRHBPCRHR2ALOX5ESR2ESR1
SCHEMBL1760592 0.78 ESR2 (0.53) PDE4BPDE4APDE4CPDE4DALOX5
SCHEMBL1535884 0.77 BACE1 (0.54) PDE4BPDE4APDE4CPDE4DALOX5
SCHEMBL4384039 0.77 PDE4B (0.47) CRHBPCRHR2PDE4BPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113549010-B Preparation and application of compound with AMPK (AMPK) agonistic activity and prodrug thereof 中国科学院上海药物研究所 2023-10-20 CN disclosed