SCHEMBL29145449

SCHEMBL29145449

Cc1nc2c(s1)C[C@H](OC(=O)NC(C)(C)C)CC2

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.41
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDK1 Q15118 1/20 0.36
TP53 P04637 3/20 0.36
POLB P06746 1/20 0.36
CCNE1 P24864 5/20 0.36
CDK2 P24941 5/20 0.36
SCN4A P35499 1/20 0.35
GSK3B P49841 1/20 0.35
MAPT P10636 4/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN3A Q9NY46 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29145446 0.88 NPC1 (0.36) NPC1RAB9ASMN1; SMN2PDK1TP53
SCHEMBL29145421 0.86 SCN4A (0.48) SCN4ASCN5ASCN3A
SCHEMBL29145459 0.85 NPC1 (0.35) NPC1RAB9ASMN1; SMN2PDK1TP53
SCHEMBL28549493 0.80 DPP4 (0.45) DPP4NPC1RAB9ASMN1; SMN2PDK1
SCHEMBL28549495 0.80 DPP4 (0.45) DPP4NPC1RAB9ASMN1; SMN2PDK1
SCHEMBL28912414 0.73 SCN4A (0.49) DPP4SCN4AGSK3BSCN5ASCN3A
SCHEMBL28912415 0.73 SCN4A (0.49) DPP4SCN4AGSK3BSCN5ASCN3A
SCHEMBL23306019 0.73 NPC1 (0.39) NPC1RAB9ASMN1; SMN2PDK1TP53
SCHEMBL27821593 0.72 THRB (0.34) DPP4SMN1; SMN2CCNE1CDK2GSK3B
SCHEMBL16286105 0.72 DPP4 (0.35) DPP4PDK1TP53POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574191-B Isoxazole heterocyclic compound and application thereof 南京圣和药业股份有限公司 2024-01-23 CN disclosed