SCHEMBL29145446

SCHEMBL29145446

CC(C)(C)NC(=O)O[C@@H]1CCc2nc(Br)sc2C1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
SCN4A P35499 1/20 0.35
TP53 P04637 5/20 0.34
MAPT P10636 4/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PDK1 Q15118 2/20 0.34
SCN3A Q9NY46 3/20 0.34
SCN5A Q14524 2/20 0.34
POLB P06746 2/20 0.34
SCN9A Q15858 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29145449 0.88 DPP4 (0.41) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL29145421 0.86 SCN4A (0.48) SCN4ASCN3ASCN5ASCN9A
SCHEMBL23306019 0.86 NPC1 (0.39) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL29145459 0.85 NPC1 (0.35) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL28560728 0.79 PDK1 (0.38) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL23306592 0.79 PDK1 (0.38) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL29145448 0.73 SCN4A (0.49) SCN4ASCN3ASCN5ASCN9A
SCHEMBL15738520 0.73 SCN4A (0.49) SCN4ASCN3ASCN5ASCN9A
SCHEMBL27821593 0.72 THRB (0.34) SMN1; SMN2
SCHEMBL25277512 0.69 EPHX1 (0.36) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574191-B Isoxazole heterocyclic compound and application thereof 南京圣和药业股份有限公司 2024-01-23 CN disclosed