SCHEMBL29145459

SCHEMBL29145459

CC(C)(C)NC(=O)O[C@H]1CCc2nc(C3CC3)sc2C1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CCNE1 P24864 8/20 0.35
CDK2 P24941 8/20 0.35
SCN4A P35499 1/20 0.34
GSK3B P49841 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
TP53 P04637 3/20 0.33
MAPT P10636 2/20 0.33
SCN5A Q14524 1/20 0.33
SCN3A Q9NY46 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
POLB P06746 1/20 0.33
PDK1 Q15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29145449 0.85 DPP4 (0.41) NPC1RAB9ASMN1; SMN2CCNE1CDK2
SCHEMBL29145446 0.85 NPC1 (0.36) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL29145421 0.84 SCN4A (0.48) SCN4ASCN5ASCN3A
SCHEMBL28565598 0.80 PDK1 (0.36) NPC1RAB9ASMN1; SMN2SCN4AHDAC9
SCHEMBL28565602 0.80 PDK1 (0.36) NPC1RAB9ASMN1; SMN2SCN4AHDAC9
SCHEMBL28912406 0.75 SCN4A (0.48) SCN4ASCN5ASCN3A
SCHEMBL28912404 0.75 SCN4A (0.48) SCN4ASCN5ASCN3A
SCHEMBL23306019 0.71 NPC1 (0.39) NPC1RAB9ASMN1; SMN2SCN4ATP53
SCHEMBL27821593 0.70 THRB (0.34) SMN1; SMN2CCNE1CDK2GSK3B
SCHEMBL25277512 0.67 EPHX1 (0.36) SMN1; SMN2CCNE1CDK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574191-B Isoxazole heterocyclic compound and application thereof 南京圣和药业股份有限公司 2024-01-23 CN disclosed