SCHEMBL2915985

SCHEMBL2915985

O=CCN1CCCOc2ccc([N+](=O)[O-])cc21

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
LMNA P02545 1/20 0.39
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
CHRNB4 P30926 4/20 0.37
CHRNA3 P32297 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37
CRHBP P24387 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHR2 Q13324 1/20 0.37
HPGD P15428 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724189 0.92 ALDH1A1 (0.43) ALDH1A1LMNAMAPTGAACHRNB4
SCHEMBL2060680 0.85 CHRNB4 (0.40) ALDH1A1LMNAMAPTGAACHRNB4
SCHEMBL2913833 0.79 MAPT (0.36) ALDH1A1MAPTGAACHRNB4CHRNA3
SCHEMBL2061015 0.79 CHRNB4 (0.46) ALDH1A1LMNAMAPTGAACHRNB4
SCHEMBL5051534 0.77 GAA (0.42) ALDH1A1LMNAMAPTGAASMN1; SMN2
SCHEMBL25607650 0.77 PIK3CD (0.43) ALDH1A1MAPTSMN1; SMN2MEN1CRHBP
SCHEMBL6368485 0.76 SMN1; SMN2 (0.43) ALDH1A1LMNAMAPTSMN1; SMN2KMT2A
SCHEMBL12404774 0.75 ALDH1A1 (0.35) ALDH1A1LMNAMAPTGAACHRNB4
SCHEMBL2910729 0.75 ESPL1 (0.38) ALDH1A1LMNAMAPTGAA
SCHEMBL2061320 0.74 ALDH1A1 (0.43) ALDH1A1LMNAMAPTGAACHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222647-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS Cephalon, Inc. (US) 2010-09-01 EP disclosed
WO-2008051547-A1 FUSED BICYCLIC DERIVATIVES OF 2,4-DIAMINOPYRIMIDINE AS ALK AND C-MET INHIBITORS CEPHALON, INC. (US) 2008-05-02 WO disclosed