SCHEMBL2917150

SCHEMBL2917150

CC(=O)N1Cc2n[nH]c(CNC(=O)c3ccco3)c2C1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
HPGD P15428 4/20 0.44
GFER P55789 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
KMT2A Q03164 2/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.41
AURKA O14965 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
GAA P10253 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
MEN1 O00255 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2922367 0.81 RAB9A (0.47) ALDH1A1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL2917155 0.81 AURKA (0.50) ALDH1A1HPGDTDP1KMT2ARAB9A
SCHEMBL2922370 0.73 AURKA (0.68) RAB9ANPC1AURKACCNA2CDK2
SCHEMBL2921958 0.67 CCNA2 (0.65) ALDH1A1HPGDKMT2ASMN1; SMN2KDM4E
SCHEMBL2916029 0.65 CCNA2 (0.41) ALDH1A1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL2921266 0.65 CCNA2 (0.63) HPGDKMT2ARAB9ANPC1AURKA
SCHEMBL5123738 0.65 ALDH1A1 (0.77) ALDH1A1HPGDKMT2ARAB9ANPC1
SCHEMBL5720799 0.64 CCNA2 (0.47) SMN1; SMN2AURKACCNA2CDK2CCNA1
SCHEMBL13074753 0.63 ALDH1A1 (0.64) ALDH1A1HPGDKMT2ARAB9ANPC1
SCHEMBL16266238 0.63 ALDH1A1 (1.00) ALDH1A1HPGDTDP1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320531-B1 BICYCLO-PYRAZOLES ACTIVE AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM PFIZER ITALIA SRL (IT) 2010-09-08 EP claimed