SCHEMBL29176352

SCHEMBL29176352

O=C(Nc1ccccc1)c1c[nH]c2cc(F)ccc12

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.57
DGAT1 O75907 1/20 0.52
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 1/20 0.51
TDO2 P48775 2/20 0.51
IDO1 P14902 1/20 0.51
HTR2C P28335 1/20 0.48
NHERF1 O14745 2/20 0.47
LMNA P02545 1/20 0.47
AVPR2 P30518 1/20 0.46
GPR27 Q9NS67 1/20 0.46
HTT P42858 1/20 0.46
KDM4E B2RXH2 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29176346 0.89 CFTR (0.60) CFTRMEN1KMT2ANPC1RAB9A
SCHEMBL28571455 0.87 NHERF1 (0.65) MEN1KMT2ANPC1RAB9ANHERF1
SCHEMBL30089269 0.87 NHERF1 (0.65) MEN1KMT2ANPC1RAB9ANHERF1
SCHEMBL30912930 0.86 P2RX1 (0.50) CFTRMEN1KMT2ANPC1RAB9A
SCHEMBL29176341 0.86 P2RX1 (0.50) CFTRMEN1KMT2ANPC1RAB9A
SCHEMBL29176366 0.83 NHERF1 (0.63) CFTRDGAT1MEN1KMT2ANPC1
SCHEMBL10260257 0.83 CFTR (0.57) CFTRDGAT1MEN1KMT2ANPC1
SCHEMBL20567516 0.83 STING1 (0.64) CFTRMEN1KMT2ANPC1RAB9A
SCHEMBL29176625 0.82 MEN1 (0.62) CFTRMEN1KMT2ANPC1RAB9A
SCHEMBL4430677 0.82 CFTR (0.80) CFTRMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024109642-A1 USE OF BENZOAZACYCLIC COMPOUND AS ALLOSTERIC MODULATOR OF β2-ADRENOCEPTOR 常州大学 2024-05-30 WO disclosed
CN-117447381-A Indole amide derivative and its application in preparing beta 2 Use of adrenoreceptor allosteric antagonist medicaments 常州大学 2024-01-26 CN disclosed