SCHEMBL29176366

SCHEMBL29176366

O=C(Nc1ccccc1)c1c[nH]c2cc(Cl)ccc12

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NHERF1 O14745 5/20 0.63
NR4A2 P43354 1/20 0.58
TMPRSS4 Q9NRS4 1/20 0.57
CFTR P13569 1/20 0.57
DGAT1 O75907 1/20 0.52
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
AVPR1A P37288 2/20 0.51
F7 P08709 1/20 0.50
F3 P13726 1/20 0.50
MAOB P27338 1/20 0.49
HRH3 Q9Y5N1 1/20 0.48
BACE1 P56817 1/20 0.47
MAPT P10636 1/20 0.47
CYP2C19 P33261 1/20 0.47
USP2 O75604 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL398244 0.91 CFTR (0.71) NHERF1NR4A2TMPRSS4CFTRMAOB
SCHEMBL29176623 0.89 NHERF1 (0.79) NHERF1NR4A2TMPRSS4CFTRF7
SCHEMBL13043506 0.86 RAB9A (0.71) NR4A2MEN1KMT2ANPC1RAB9A
SCHEMBL31448058 0.84 NPC1 (0.53) NHERF1NR4A2TMPRSS4CFTRMEN1
SCHEMBL29176352 0.83 CFTR (0.57) NHERF1CFTRDGAT1MEN1KMT2A
SCHEMBL10260257 0.83 CFTR (0.57) NHERF1CFTRDGAT1MEN1KMT2A
SCHEMBL20567521 0.83 STING1 (0.64) NHERF1CFTRMEN1KMT2ANPC1
SCHEMBL18229436 0.83 CFTR (0.71) NHERF1NR4A2TMPRSS4CFTRF7
SCHEMBL30695128 0.82 NHERF1 (0.65) NHERF1CFTRMEN1KMT2ANPC1
SCHEMBL29176615 0.82 NHERF1 (0.65) NHERF1CFTRMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024109642-A1 USE OF BENZOAZACYCLIC COMPOUND AS ALLOSTERIC MODULATOR OF β2-ADRENOCEPTOR 常州大学 2024-05-30 WO disclosed
CN-117447381-A Indole amide derivative and its application in preparing beta 2 Use of adrenoreceptor allosteric antagonist medicaments 常州大学 2024-01-26 CN disclosed