SCHEMBL29176830

SCHEMBL29176830

CCOC(=O)C(C(=O)OCC)c1cccc(-c2noc(C(C)C)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 2/20 0.49
KCNT1 Q5JUK3 1/20 0.43
NPY2R P49146 1/20 0.42
S1PR3 Q99500 2/20 0.42
HTT P42858 2/20 0.42
BMP1 P13497 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
TP53 P04637 1/20 0.41
KCNH2 Q12809 1/20 0.41
S1PR1 P21453 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTPN1 P18031 1/20 0.40
ACACB O00763 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29176878 0.90 KCNH2 (0.42) AAK1KCNT1S1PR3HTTBMP1
SCHEMBL29176877 0.87 L3MBTL1 (0.56) HTTTP53KCNH2MAPTMAPK1
SCHEMBL29176874 0.85 KCNH2 (0.48) HTTNPSR1TP53KCNH2MAPT
SCHEMBL29176870 0.85 NPC1 (0.47) S1PR3HTTNPSR1TP53S1PR1
SCHEMBL29176879 0.84 KCNH2 (0.42) AAK1HTTBMP1NPSR1TP53
SCHEMBL30817786 0.84 S1PR3 (0.46) NPY2RS1PR3HTTNPSR1S1PR1
SCHEMBL29176876 0.84 S1PR3 (0.46) NPY2RS1PR3HTTNPSR1S1PR1
SCHEMBL30817792 0.83 S1PR3 (0.43) AAK1KCNT1NPY2RS1PR3HTT
SCHEMBL29176836 0.83 S1PR3 (0.43) AAK1KCNT1NPY2RS1PR3HTT
SCHEMBL29176835 0.82 HDAC4 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117720535-A Pyrido [1,2-a ] pyrimidine mesoionic derivative containing 1,2, 4-oxadiazole structure, and preparation and application thereof 贵州大学 2024-03-19 CN disclosed